利血平

英文名称：Reserpine
CAS号：50-55-5
分析标准品,≥99.5%
分子式 C33H40N2O9 分子量608.68

基本信息:

密度1.32
溶解性 Soluble in DMSO (100 mM), chloroform (10 mg/ml), water (<1 mg/ml at 25° C), and ethanol (<1 mg/ml at 25° C).
存贮条件 储存温度2-8°C
描述
产品介绍 Reserpine has displayed a capacity to inhibit the transport of biogenic amines into synaptic vesicles and adrenal chromaffin granules. The mechanism behind this inhibition has been illuminated as an irreversible binding to the vesicular amine transporter. Furthermore, Reserpine has been reported to interfere with dopamine transporter activity and potently inhibit synaptosomal dopamine uptake. Reserpine is an inhibitor of VMAT 2.
别名 蛇根碱;血安平;蛇根草素;Serpalan; Serpasil; Hiserpia; Serpanray; Serpivite; Apoplon;3,4,5-Trimethoxybenzoyl methyl reserpate; (3β, 16β, 17α, 18β, 20α)-11,17-Dimethoxy-18-[(3,4,5-trimethoxybenzoyl)oxy]yohimban-16-carboxylic acid methyl ester
生化机理 抑制儿茶酚胺(catecholamines)和5-羟色胺（serotonin）的吸收。
应用 An inhibitor of transport of biogenic amines into adrenal chromaffin granules